gene_symbol
TACSTD2
hgnc_id
HGNC:11530
binding_type
antigen recognition
cytotoxicity
YES
cytotoxicity_type
DIRECT
cytotoxicity_mechanism
Anti–TROP-2 antibody–drug conjugate binds TROP-2, is internalized, and releases SN-38, a topoisomerase I inhibitor, causing DNA damage and apoptosis in target cells (with potential bystander effect).
enzyme_product
Off
epitope
On
variant
Off
isoform
Off
hla_specific
Off
gated
Off
other_modifier
ADC antibody antigen target
trial_id_tar_ref
drug_id_tar_ref
disease_id_tar_ref
nct_id_tar_ref
NCT06328387
disease_id_num_tar_ref
1246
drug_id_num_tar_ref
3377