gene_symbol
EGFR
hgnc_id
HGNC:3236
binding_type
antigen recognition
cytotoxicity
YES
cytotoxicity_type
DIRECT
cytotoxicity_mechanism
ADC binds EGFR, is internalized, and releases MMAE, which inhibits tubulin polymerization leading to G2/M arrest and apoptosis of EGFR-expressing cells.
enzyme_product
On
epitope
Off
variant
Off
isoform
Off
hla_specific
Off
gated
Off
other_modifier
Antibody target (becotatug moiety)
trial_id_tar_ref
drug_id_tar_ref
disease_id_tar_ref
nct_id_tar_ref
NCT06530914
disease_id_num_tar_ref
1872
drug_id_num_tar_ref
4979