gene_symbol
FOLH1
hgnc_id
HGNC:3788
binding_type
receptor ligand recognition
cytotoxicity
YES
cytotoxicity_type
DIRECT
cytotoxicity_mechanism
PSMA-binding Lu-177 radioligand is internalized and emits β-particles that cause DNA double-strand breaks, killing PSMA-positive cells (with beta crossfire to nearby cells).
enzyme_product
Off
epitope
Off
variant
Off
isoform
Off
hla_specific
Off
gated
Off
other_modifier
Membrane enzyme target; ligand binding leads to internalization
trial_id_tar_ref
drug_id_tar_ref
disease_id_tar_ref
nct_id_tar_ref
NCT05682443
disease_id_num_tar_ref
3968
drug_id_num_tar_ref
10717