gene_symbol
EGFR
hgnc_id
HGNC:3236
binding_type
other
cytotoxicity
NO
cytotoxicity_type
DIRECT
cytotoxicity_mechanism
Not killed. Lazertinib is a mutant‑selective EGFR TKI with minimal activity against wild‑type EGFR; cytotoxicity occurs only in EGFR‑mutant cells via direct blockade of EGFR signaling leading to apoptosis.
enzyme_product
On
epitope
Off
variant
Off
isoform
Off
hla_specific
Off
gated
Off
other_modifier
Covalent binding at Cys797 with minimal inhibitory activity versus wild-type EGFR
trial_id_tar_ref
drug_id_tar_ref
disease_id_tar_ref
nct_id_tar_ref
NCT05663866
disease_id_num_tar_ref
4112
drug_id_num_tar_ref
11101