gene_symbol
NTRK3
hgnc_id
HGNC:8033
binding_type
other
cytotoxicity
YES
cytotoxicity_type
DIRECT
cytotoxicity_mechanism
Entrectinib directly inhibits TRKC (NTRK3) kinase activity, shutting down MAPK/PI3K survival signaling in TRKC-driven tumor cells and inducing apoptosis.
enzyme_product
On
epitope
Off
variant
Off
isoform
Off
hla_specific
Off
gated
Off
other_modifier
receptor tyrosine kinase (TrkC); often activated by NTRK3 gene fusions
trial_id_tar_ref
drug_id_tar_ref
disease_id_tar_ref
nct_id_tar_ref
NCT05862285
disease_id_num_tar_ref
5703
drug_id_num_tar_ref
15497